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In this experiment, we established the normal albumin concentration of a healthy adult (600 μ M) or a low-albumin state indicating marked liver hypofunction (100 μ M) on a cell membrane plate, and evaluated the cell membrane permeability of the probe agents. The cell membrane permeability of phenytoin or valproate depended on the concentration of albumin. Probe agent site-I and -II inhibitors, bucolome and oleic acid, respectively, increased the cell membrane permeability. In the future, the cell membrane permeability of probe agents should be further investigated to estimate the tissue transfer of agents based on various laboratory data (albumin, free fatty acids, uremic toxins, and bilirubin).","subitem_description_type":"Other"}]},"item_1_identifier_registration":{"attribute_name":"ID登録","attribute_value_mlt":[{"subitem_identifier_reg_text":"10.15069/00000907","subitem_identifier_reg_type":"JaLC"}]},"item_1_source_id_13":{"attribute_name":"雑誌書誌ID","attribute_value_mlt":[{"subitem_source_identifier":"AA11490417","subitem_source_identifier_type":"NCID"}]},"item_1_text_10":{"attribute_name":"著者所属(英)","attribute_value_mlt":[{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Medical Engineering, College of Health Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Graduate School of Medical Science, Kanazawa University"},{"subitem_text_language":"en","subitem_text_value":"Graduate School of Medical Science, Kanazawa University"}]},"item_1_text_9":{"attribute_name":"著者所属(日)","attribute_value_mlt":[{"subitem_text_value":"九州保健福祉大学薬学部薬学科"},{"subitem_text_value":"九州保健福祉大学薬学部薬学科"},{"subitem_text_value":"九州保健福祉大学薬学部薬学科"},{"subitem_text_value":"九州保健福祉大学薬学部薬学科"},{"subitem_text_value":"九州保健福祉大学薬学部薬学科"},{"subitem_text_value":"九州保健福祉大学保健科学部臨床工学科"},{"subitem_text_value":"金沢大学大学院医学研究科"},{"subitem_text_value":"金沢大学大学院医学研究科"}]},"item_files":{"attribute_name":"ファイル情報","attribute_type":"file","attribute_value_mlt":[{"accessrole":"open_date","date":[{"dateType":"Available","dateValue":"2009-03-01"}],"displaytype":"simple","filename":"30 研究紀要 10号 徳永.pdf","filesize":[{"value":"674.4 kB"}],"format":"application/pdf","licensetype":"license_11","mimetype":"application/pdf","url":{"label":"30 研究紀要 10号 徳永","url":"https://phoenix.repo.nii.ac.jp/record/915/files/30 研究紀要 10号 徳永.pdf"},"version_id":"5da98da2-7767-4ba3-a561-30dc1f86af08"}]},"item_keyword":{"attribute_name":"キーワード","attribute_value_mlt":[{"subitem_subject":"薬学的分布診断法","subitem_subject_scheme":"Other"},{"subitem_subject":"細胞膜プレート","subitem_subject_scheme":"Other"},{"subitem_subject":"プローブ薬物","subitem_subject_scheme":"Other"},{"subitem_subject":"ヒト血清アルブミン","subitem_subject_scheme":"Other"},{"subitem_subject":"蛋白結合","subitem_subject_scheme":"Other"},{"subitem_subject":"pharmaceutical distribution diagnostic method","subitem_subject_language":"en","subitem_subject_scheme":"Other"},{"subitem_subject":"cell membrane plate","subitem_subject_language":"en","subitem_subject_scheme":"Other"},{"subitem_subject":"probe agent","subitem_subject_language":"en","subitem_subject_scheme":"Other"},{"subitem_subject":"human serum albumin","subitem_subject_language":"en","subitem_subject_scheme":"Other"},{"subitem_subject":"protein binding","subitem_subject_language":"en","subitem_subject_scheme":"Other"}]},"item_language":{"attribute_name":"言語","attribute_value_mlt":[{"subitem_language":"jpn"}]},"item_resource_type":{"attribute_name":"資源タイプ","attribute_value_mlt":[{"resourcetype":"departmental bulletin paper","resourceuri":"http://purl.org/coar/resource_type/c_6501"}]},"item_title":"細胞膜プレートを使用したサイトプローブ薬物の細胞膜透過性に関する基礎的検討","item_titles":{"attribute_name":"タイトル","attribute_value_mlt":[{"subitem_title":"細胞膜プレートを使用したサイトプローブ薬物の細胞膜透過性に関する基礎的検討"},{"subitem_title":"Basic examination of the cell membrane permeability of site probe agents using a cell membrane plate","subitem_title_language":"en"}]},"item_type_id":"1","owner":"3","path":["52"],"pubdate":{"attribute_name":"公開日","attribute_value":"2009-03-25"},"publish_date":"2009-03-25","publish_status":"0","recid":"915","relation_version_is_last":true,"title":["細胞膜プレートを使用したサイトプローブ薬物の細胞膜透過性に関する基礎的検討"],"weko_creator_id":"3","weko_shared_id":3},"updated":"2024-04-19T07:10:59.361742+00:00"}