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濃度に有意な差はみられなかった。また肝癌ラットを使用したin vivo 実験系において、L-cysteine を併用したcisplatin の肝動注はcisplatin のみの投与に比べ、腫瘍増殖率が抑えられる傾向であることを示した。さらに肝組織中における腫瘍部と非腫瘍部におけるcisplatin 濃度において、L-cysteine 併用により腫瘍部と非腫瘍部に有意な差を認めることができた (p<0.01)。以上の結果より、L-cysteine の併用はcisplatin の肝動注療法へ応用できると考えられる。","subitem_description_type":"Other"}]},"item_1_description_12":{"attribute_name":"抄録(英)","attribute_value_mlt":[{"subitem_description":"Covalent binding is involved in the protein binding of cisplatin. L-cysteine reduces the covalent binding of cisplatin. We investigated hepatic arterial infusion therapy with cisplatin using protein binding inhibition. In the present experiment, the pharmacokinetics and antineoplastic effects of cisplatin combined with L-cysteine in male Donryu rats were investigated. As a result, no significant difference was noted in the total and free concentrations of cisplatin combined with L-cysteine. In an in vivo experiment using rats with liver cancer, the hepatic arterial infusion of cisplatin combined with L-cysteine showed that it was the tendency that tumor growth rate was inhibited in comparison with administration only for cisplatin. In addition, concentrations of cisplatin increased significantly between tumor and non-tumor regions in liver tissue when combined with L-cysteine (p<0.01). Thus, L-cysteine can be combined with cisplatin for hepatic arterial infusion therapy.","subitem_description_type":"Other"}]},"item_1_identifier_registration":{"attribute_name":"ID登録","attribute_value_mlt":[{"subitem_identifier_reg_text":"10.15069/00000933","subitem_identifier_reg_type":"JaLC"}]},"item_1_source_id_13":{"attribute_name":"雑誌書誌ID","attribute_value_mlt":[{"subitem_source_identifier":"AA11490417","subitem_source_identifier_type":"NCID"}]},"item_1_text_10":{"attribute_name":"著者所属(英)","attribute_value_mlt":[{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmacy, University Hospital of Medicine, Tokyo Medical and Dental University"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutics, Faculty of Pharmaceutical Sciences, Kobe Gakuin University"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmaceutics, Faculty of Pharmaceutical Sciences, Kobe Gakuin University"},{"subitem_text_language":"en","subitem_text_value":"Department of Diagnostic Radiology, Kumamoto University Graduate School of Medical and Pharmaceutical Sciences"},{"subitem_text_language":"en","subitem_text_value":"Faculty of Health Sciences, Institute of Medical, Pharmaceutical and Health Sciences, Kanazawa University"},{"subitem_text_language":"en","subitem_text_value":"Faculty of Health Sciences, Institute of Medical, Pharmaceutical and Health Sciences, Kanazawa University"},{"subitem_text_language":"en","subitem_text_value":"Department of Pharmacy, Faculty of Medicine, University of Miyazaki 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