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細胞膜プレートを使用したサイトプローブ薬物の細胞膜透過性に関する基礎的検討
名前 / ファイル | ライセンス | アクション |
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30 研究紀要 10号 徳永 (674.4 kB)
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Item type | 紀要論文(ELS) / Departmental Bulletin Paper(1) | |||||||||||||||||||||||||||
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公開日 | 2009-03-25 | |||||||||||||||||||||||||||
タイトル | ||||||||||||||||||||||||||||
タイトル | 細胞膜プレートを使用したサイトプローブ薬物の細胞膜透過性に関する基礎的検討 | |||||||||||||||||||||||||||
タイトル | ||||||||||||||||||||||||||||
言語 | en | |||||||||||||||||||||||||||
タイトル | Basic examination of the cell membrane permeability of site probe agents using a cell membrane plate | |||||||||||||||||||||||||||
言語 | ||||||||||||||||||||||||||||
言語 | jpn | |||||||||||||||||||||||||||
キーワード | ||||||||||||||||||||||||||||
主題Scheme | Other | |||||||||||||||||||||||||||
主題 | 薬学的分布診断法 | |||||||||||||||||||||||||||
キーワード | ||||||||||||||||||||||||||||
主題Scheme | Other | |||||||||||||||||||||||||||
主題 | 細胞膜プレート | |||||||||||||||||||||||||||
キーワード | ||||||||||||||||||||||||||||
主題Scheme | Other | |||||||||||||||||||||||||||
主題 | プローブ薬物 | |||||||||||||||||||||||||||
キーワード | ||||||||||||||||||||||||||||
主題Scheme | Other | |||||||||||||||||||||||||||
主題 | ヒト血清アルブミン | |||||||||||||||||||||||||||
キーワード | ||||||||||||||||||||||||||||
主題Scheme | Other | |||||||||||||||||||||||||||
主題 | 蛋白結合 | |||||||||||||||||||||||||||
キーワード | ||||||||||||||||||||||||||||
言語 | en | |||||||||||||||||||||||||||
主題Scheme | Other | |||||||||||||||||||||||||||
主題 | pharmaceutical distribution diagnostic method | |||||||||||||||||||||||||||
キーワード | ||||||||||||||||||||||||||||
言語 | en | |||||||||||||||||||||||||||
主題Scheme | Other | |||||||||||||||||||||||||||
主題 | cell membrane plate | |||||||||||||||||||||||||||
キーワード | ||||||||||||||||||||||||||||
言語 | en | |||||||||||||||||||||||||||
主題Scheme | Other | |||||||||||||||||||||||||||
主題 | probe agent | |||||||||||||||||||||||||||
キーワード | ||||||||||||||||||||||||||||
言語 | en | |||||||||||||||||||||||||||
主題Scheme | Other | |||||||||||||||||||||||||||
主題 | human serum albumin | |||||||||||||||||||||||||||
キーワード | ||||||||||||||||||||||||||||
言語 | en | |||||||||||||||||||||||||||
主題Scheme | Other | |||||||||||||||||||||||||||
主題 | protein binding | |||||||||||||||||||||||||||
資源タイプ | ||||||||||||||||||||||||||||
資源タイプ識別子 | http://purl.org/coar/resource_type/c_6501 | |||||||||||||||||||||||||||
資源タイプ | departmental bulletin paper | |||||||||||||||||||||||||||
ID登録 | ||||||||||||||||||||||||||||
ID登録 | 10.15069/00000907 | |||||||||||||||||||||||||||
ID登録タイプ | JaLC | |||||||||||||||||||||||||||
ページ属性 | ||||||||||||||||||||||||||||
内容記述タイプ | Other | |||||||||||||||||||||||||||
内容記述 | P(論文) | |||||||||||||||||||||||||||
著者名(日) |
徳永, 仁
× 徳永, 仁
WEKO
1014
× 高村, 徳人
WEKO
1013
× 緒方, 賢次
WEKO
1012
× 吉田, 裕樹
WEKO
5925
× 永田, 将司× 近藤, 照義× 西尾, 豊隆× 川井, 恵一 |
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著者名よみ |
トクナガ, ジン
× トクナガ, ジン× タカムラ, ノリト× オガタ, ケンジ× ヨシダ, ヒロキ× ナガタ, マサシ× コンドウ, テルヨシ× ニシオ, トヨタカ× カワイ, ケイイチ |
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著者名(英) |
TOKUNAGA, Jin
× TOKUNAGA, Jin× TAKAMURA, Norito× OGATA, Kenji× YOSHIDA, Hiroki× NAGATA, Masashi× KONDO, Teruyoshi× NISHIO, Toyotaka× KAWAI, Keiichi |
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著者所属(日) | ||||||||||||||||||||||||||||
九州保健福祉大学薬学部薬学科 | ||||||||||||||||||||||||||||
著者所属(日) | ||||||||||||||||||||||||||||
九州保健福祉大学薬学部薬学科 | ||||||||||||||||||||||||||||
著者所属(日) | ||||||||||||||||||||||||||||
九州保健福祉大学薬学部薬学科 | ||||||||||||||||||||||||||||
著者所属(日) | ||||||||||||||||||||||||||||
九州保健福祉大学薬学部薬学科 | ||||||||||||||||||||||||||||
著者所属(日) | ||||||||||||||||||||||||||||
九州保健福祉大学薬学部薬学科 | ||||||||||||||||||||||||||||
著者所属(日) | ||||||||||||||||||||||||||||
九州保健福祉大学保健科学部臨床工学科 | ||||||||||||||||||||||||||||
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金沢大学大学院医学研究科 | ||||||||||||||||||||||||||||
著者所属(日) | ||||||||||||||||||||||||||||
金沢大学大学院医学研究科 | ||||||||||||||||||||||||||||
著者所属(英) | ||||||||||||||||||||||||||||
en | ||||||||||||||||||||||||||||
Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare | ||||||||||||||||||||||||||||
著者所属(英) | ||||||||||||||||||||||||||||
en | ||||||||||||||||||||||||||||
Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare | ||||||||||||||||||||||||||||
著者所属(英) | ||||||||||||||||||||||||||||
en | ||||||||||||||||||||||||||||
Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare | ||||||||||||||||||||||||||||
著者所属(英) | ||||||||||||||||||||||||||||
en | ||||||||||||||||||||||||||||
Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare | ||||||||||||||||||||||||||||
著者所属(英) | ||||||||||||||||||||||||||||
en | ||||||||||||||||||||||||||||
Department of Pharmaceutical Sciences, School of Pharmaceutical Sciences, Kyushu University of Health and Welfare | ||||||||||||||||||||||||||||
著者所属(英) | ||||||||||||||||||||||||||||
en | ||||||||||||||||||||||||||||
Department of Medical Engineering, College of Health Sciences, Kyushu University of Health and Welfare | ||||||||||||||||||||||||||||
著者所属(英) | ||||||||||||||||||||||||||||
en | ||||||||||||||||||||||||||||
Graduate School of Medical Science, Kanazawa University | ||||||||||||||||||||||||||||
著者所属(英) | ||||||||||||||||||||||||||||
en | ||||||||||||||||||||||||||||
Graduate School of Medical Science, Kanazawa University | ||||||||||||||||||||||||||||
抄録(英) | ||||||||||||||||||||||||||||
内容記述タイプ | Other | |||||||||||||||||||||||||||
内容記述 | Drug efficacy depends on the amount of a preparation reaching the target tissue (grade of tissue transfer). In this experiment, we established the normal albumin concentration of a healthy adult (600 μ M) or a low-albumin state indicating marked liver hypofunction (100 μ M) on a cell membrane plate, and evaluated the cell membrane permeability of the probe agents. The cell membrane permeability of phenytoin or valproate depended on the concentration of albumin. Probe agent site-I and -II inhibitors, bucolome and oleic acid, respectively, increased the cell membrane permeability. In the future, the cell membrane permeability of probe agents should be further investigated to estimate the tissue transfer of agents based on various laboratory data (albumin, free fatty acids, uremic toxins, and bilirubin). | |||||||||||||||||||||||||||
雑誌書誌ID | ||||||||||||||||||||||||||||
収録物識別子タイプ | NCID | |||||||||||||||||||||||||||
収録物識別子 | AA11490417 | |||||||||||||||||||||||||||
書誌情報 |
九州保健福祉大学研究紀要 en : Journal of Kyushu University of Health and Welfare 巻 10, p. 193-199, 発行日 2009-03 |